型号:
产品价格:电议      采购度:1604      原产地:美洲
发布时间:2021/7/21 16:31:51 所属地区:上海 上海市
简要描述:
Angiotensin II 5-valine 是血管紧张素受体 (angiotensin receptor) 的激动剂。
标签:Valine angiotensin II
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CAS No. : 58-49-1
MCE 站:Angiotensin II 5-valine
产品活性:Angiotensin II 5-valine 是血管紧张素受体 (angiotensin receptor) 的激动剂。
研究领域:GPCR/G Protein
作用靶点:Angiotensin Receptor
In Vivo: By day 12, systolic blood pressure (SBP) increases significantly in Angiotensin II 5-valine infused rats (197±7 mm Hg). As shown, the development of hypertension in ANG II infused rats is prevented by losartan treatment. Blood and kidney samples are harvested, subjected to HPLC to separate Angiotensin II 5-valine (exogenous) from Ile5-ANG II (endogenous) and the fractions are measured by radioimmunoassay. In the Angiotensin II 5-valine infused rats treated with losartan, total plasma ANG II levels are elevated to a greater extent than in rats not treated with losartan (289±20 v 119±14 fmol/mL). However, losartan markedly decrease by 88% the enhancement of intrarenal Val5-ANG II content that occurred in the rats infused with Val5-ANG II alone.
相关产品:Drug Repurposing Compound Library Plus | FDA-Approved Drug Library Plus | Bioactive Compound Library Plus | GPCR/G Protein Compound Library | FDA-Approved Drug Library | Anti-Cancer Compound Library | Peptidomimetic Library | Drug Repurposing Compound Library | Endocrinology Compound Library | Neurotransmitter Receptor Compound Library | FDA Approved & Pharmacopeial Drug Library | Angiotensin II human | Losartan | A 779 | Telmisartan | PD 123319 ditrifluoroacetate | AVE 0991 | Valsartan | Olmesartan | Tranilast | YS-49 | Irbesartan | Candesartan | CGP-42112 | Olodanrigan | Sparsentan | C-Type Natriuretic Peptide (CNP) (1-22), human | Azilsartan medoxomil | Eprosartan mesylate | Angiotensin (1-7) (acetate) | Fimasartan | Tasosartan | Angiotensin II (3-8), human TFA | Brain Natriuretic Peptide (1-32), rat acetate
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更新时间:2024/1/2 10:14:03
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