型号:
产品价格:电议      采购度:1605      原产地:美洲
发布时间:2021/7/26 23:44:26 所属地区:上海 上海市
简要描述:
Azelastine hydrochloride 属于抗组胺剂,是一种有效的选择性组胺 1 (H1) 拮抗剂。Azelastine hydrochloride 可用于过敏性鼻炎、哮喘、糖尿病高脂血症和 SARS-CoV-2 的研究。
标签:Astelin
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CAS No. : 79307-93-0
MCE 站:Azelastine hydrochloride
产品活性:Azelastine hydrochloride 属于抗组胺剂,是一种有效的选择性组胺 1 (H1) 拮抗剂。Azelastine hydrochloride 可用于过敏性鼻炎、哮喘、糖尿病高脂血症和 SARS-CoV-2 的研究。
研究领域:GPCR/G Protein | Neuronal Signaling | Immunology/Inflammation | Anti-infection
作用靶点:Histamine Receptor | SARS-CoV
In Vitro: Azelastine hydrochloride can significantly inhibit HNEpC proliferation, and therefore, be helpful in against airway remodeling.
In Vivo: Azelastine hydrochloride (4 mg/kg; p.o.; daily; for 8 weeks) significantly reduces blood glucose, HbA1c and serum alkaline phosphatase (ALP), osteocalcin and downregulates apolipoprotein B in diabetic hyperlipidemic rats model.
Azelastine hydrochloride (4 mg/kg; p.o.; daily; for 8 weeks) improves the lipid profile (LDL-c decrease and HDL-c increase) in diabetic hyperlipidemic rats model.
Azelastine hydrochloride (4 mg/kg; p.o.; daily; for 8 weeks) attenuates calcium deposition and aortic calcification in diabetic hyperlipidemic rats model.
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更新时间:2024/1/2 10:16:09
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