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产品价格:电议      采购度:1613      原产地:美洲
发布时间:2021/8/2 20:55:56 所属地区:上海 上海市
简要描述:
Tacrine hydrochloride (hydrate) 是乙酰胆碱酯酶 (AChE) 和丁酰胆碱酯酶 (BChE) 的抑制剂,其 IC50 值分别为 31 nM 和 nM。
标签:THA
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CAS No. : 206658-92-6
MCE 站:Tacrine hydrochloride (hydrate)
产品活性:Tacrine hydrochloride (hydrate) 是乙酰胆碱酯酶 (AChE) 和丁酰胆碱酯酶 (BChE) 的抑制剂,其 IC50 值分别为 31 nM 和 25.6 nM。
研究领域:Neuronal Signaling
作用靶点:AChE
In Vitro: Tacrine hydrochloride (hydrate) (12.5 to 37.5 nM) inhibits venom acetylcholinesterase as well as human serum butyrylcholinesterase in a concentration-dependent manner. The IC50 is 31 nM for snake venom AChE and 25.6 nM for human BChE.
In Vivo: Pretreatment with Tacrine hydrochloride (hydrate) also modifies absolute levels of cocaine self-administration during reacquisition. Body weight declines approximately one-half percent over four days of treatment with intravenous Tacrine hydrochloride (hydrate). Delivery of Tacrine hydrochloride (hydrate) by osmotic pump does not alter either linear- or repeated- cocaine-induced locomotor activity. There is no significant main effect or interaction with Tacrine hydrochloride (hydrate) treatment on active lever responding during reinstatement. Post hoc comparisons indicate that rats self-administering cocaine has significantly lower alkaline phosphatase levels, relative to TTacrine hydrochloride (hydrate)- but not saline- treated rats evaluated by conditioned-place preference.
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更新时间:2024/1/2 10:17:44
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